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BRAFi :

•

Dabrafenib

•

Vemurafenib

•

Encorafenib*

MEKi :

•

Trametinib

•

Cobimetinib

•

Binimetinib*

*Not approved yet

Singh Cancer 2016 ; 15;8(1) : 1-15

Biological rationale for MEK/BRAF inhibitors

combination

BRAFi